Site‐Selective Trifluoromethylation Reactions of Oligopeptides
نویسندگان
چکیده
منابع مشابه
Investigations into Transition-Metal-Catalyzed Arene Trifluoromethylation Reactions Transition-Metal-Catalyzed Arene Trifluoromethylation Reactions
Trifluoromethyl-substituted arenes and heteroarenes are widely prevalent in pharmaceuticals and agrochemicals. As a result, the development of practical methods for the formation of aryl–CF3 bonds has become an active field of research. Over the past five years, transition-metal-catalyzed cross-coupling between aryl–X (X = halide, organometallic, or H) and various ‘CF3’ reagents has emerged as ...
متن کاملInvestigations into Transition Metal Catalyzed Arene Trifluoromethylation Reactions.
Trifluoromethyl-substituted arenes and heteroarenes are widely prevalent in pharmaceuticals and agrochemicals. As a result, the development of practical methods for the formation of aryl-CF3 bonds has become an active field of research. Over the past five years, transition metal catalyzed cross-coupling between aryl-X (X = halide, organometallic, or H) and various "CF3" reagents has emerged as ...
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Hypervalent iodine compounds are privileged reagents in organic synthesis because of their exceptional reactivity. Among these compounds, cyclic derivatives stand apart because of their enhanced stability. They have been widely used as oxidants, but their potential for functional-group transfer has only begun to be investigated recently. The use of benziodoxol(on)es for trifluoromethylation (To...
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ژورنال
عنوان ژورنال: Asian Journal of Organic Chemistry
سال: 2020
ISSN: 2193-5807,2193-5815
DOI: 10.1002/ajoc.202000170